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The main metabolic pathway of domperidone is through CYP3A4In vitro data suggest that the concomitant use of drugs that significantly inhibit this enzyme may result in increased plasma levels of domperidone.

It was found there have been 342 reports of serious side effects and 57 people known to have died from heart problems while taking domperidone.

Motilium is contraindicated in moderate or severe hepatic impairmentsee section 4.3Dose modification in mild hepatic impairment is however not neededsee section 5.2

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